Erowid.org: Erowid Reference 9086 : Fentanyl analogues with a modified propanamido group as potential affinity labels: synthesis and in vivo activity : Essawi MY

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Essawi MY. “Fentanyl analogues with a modified propanamido group as potential affinity labels: synthesis and in vivo activity”. Pharmazie. 1999 Apr 28;54(4):307-8. <a name="ref">Essawi MY.</a> <a href="/references/9086">"Fentanyl analogues with a modified propanamido group as potential affinity labels: synthesis and in vivo activity"</a> <i>Pharmazie</i>. 1999 Apr 28;54(4):307-8.
Text Abstract (this page) Full Text - English (private) Show Articles by Essawi MY Article IDs Erowid RefID: 9086 PubMedID: 10234745 Collections Hofmann Collection MDMA Collection All References	Abstract This report describes the synthesis and analgesic activity (hot-plate test) of potential affinity labels of the mu-opioid fentanyl (1) [3]. In these derivatives (2-5), the propanamido group of fentanyl was modified to include an electrophilic center which may interact with a receptor nucleophile.
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